Sunrise Malegra FXT 10 tabs (100 + 40 mg/tab)

Sildenafil

Sildenafil, commonly known as Sildenafil, is a potent PDE5 inhibitor famously marketed as Viagra. Here’s a summary of its key aspects.

Mechanism of Action

• This medication effectively blocks phosphodiesterase type 5, enhancing levels of cyclic guanosine monophosphate (cGMP) during sexual stimulation, which promotes relaxation in penile blood vessels leading to increased blood flow and erection.
• It enables both the achievement and maintenance of an erection.

Ενδείξεις

• Primarily utilized to treat erectile dysfunction in men.
• Also prescribed to address arterial hypertension under the brand name Revatio.

Onset of Action

• Typically, the effects of sildenafil manifest within 30 minutes post-administration, although it may take up to 1 hour for some individuals.

Duration of Action

• Its effectiveness lasts approximately 4 to 5 hours, facilitating erection stability during this timeframe.

Δοσολογία

• The standard initial dosage is 50 mg, adjustable based on individual tolerance and therapeutic needs.
• Doses should be consumed around 30 minutes to 1 hour prior to sexual activity.

Παρενέργειες

• Common adverse effects may include headache, facial flushing, digestive issues (nausea, diarrhea), visual disturbances, elevated blood pressure, and, in rare cases, hearing loss.

Αντενδείξεις

• Avoid concurrent use with nitrates, such as nitroglycerin, due to risks of significant hypotension. Contraindicated in individuals with severe cardiovascular conditions or recent serious heart events.

Φλουοξετίνη

Fluoxetine, often recognized as Φλουοξετίνη or Prozac, belongs to the class of selective serotonin reuptake inhibitors (SSRIs). Below are its fundamental characteristics.

Mechanism of Action

• Fluoxetine enhances serotonin levels in the brain by inhibiting its reuptake in nerve cells, increasing serotonin’s availability for receptor engagement.

Ενδείξεις

• Indicated for the treatment of depressive disorders.
• Also beneficial for obsessive-compulsive disorder (OCD), eating disorders (like bulimia nervosa), and occasionally for generalized anxiety disorder (GAD).

Onset of Action

• Fluoxetine typically takes several weeks to achieve its full therapeutic impact, with gradual improvements in mood, anxiety levels, and behavior.

Δοσολογία

The dosage of fluoxetine varies by condition:

• For depression, initiate with 20 mg daily, adjusting as necessary.
• For OCD, the starting dose ranges from 20 mg to 60 mg daily.
• For bulimia nervosa, begin with approximately 60 mg per day.

Παρενέργειες

Potential side effects include:

• Νευρικότητα
• Insomnia or excessive drowsiness
• Gastrointestinal issues (nausea, diarrhea)
• Απώλεια της όρεξης
• Αυξημένη irritability
• Απώλεια βάρους
• Altered sexual function

Αντενδείξεις

• Should not be taken alongside MAO inhibitors to prevent serious interactions that may lead to serotonin syndrome.
• Contraindicated for patients with severe liver issues or known allergies to fluoxetine.