Hilma Biocare Testosterone Undecanoate 10 ml vial (250 mg/ml)

Testosterone Undecanoate

Is a long-acting Testosterone formulation specifically designed for individuals with low or absent hormone levels. Unlike traditional esters, this formulation is available as an oral pill, with an injectable option found in Europe. The unique undecanoate ring allows the testosterone to bypass hepatic metabolism. In North America, the oral form is accessible through underground markets. Despite its advanced formulation, many bodybuilders report minimal effectiveness, often noting a lack of noticeable results.

Pharmacology

The human body naturally produces sex hormones like testosterone, essential for the development of secondary sexual characteristics, including the growth of the prostate, testes, and body hair. A deficiency in testosterone therapy is often indicated for individuals with hormone insufficiencies or infertility issues.

Indications for Use

This formulation is indicated for conditions in men characterized by insufficient testosterone production, including:

• Primary testicular insufficiency
• Pituitary failure to secrete Gonadotropins

Bodybuilding

Testosterone and its derivatives are prevalent among athletes and bodybuilders seeking to enhance physical performance and mental drive. However, many users report limited benefits, with slight weight gain being the only consistent effect. Determining the efficacy can be challenging due to the concurrent use of various substances. Testosterone possesses moderate anabolic properties alongside robust androgenic effects.
Andriol is consumed orally in doses ranging from 25-200 mg per day. Yet, most bodybuilders observe minimal results even at higher dosages, close to 400 mg/day. Extended usage of over 4-6 weeks may result in slight increases in muscle mass, contingent on a caloric-rich diet. It is essential to note that testosterone converts to estrogen in adipose tissue, elevating the risk of gynecomastia and fluid retention. To mitigate these risks, many bodybuilders incorporate Arimidex or tamoxifen during cycles.
Excessive testosterone use suppresses the body’s natural release through pituitary feedback loops, potentially impairing spermatogenesis. A gradual tapering off of the drug is recommended to allow recovery of the hypothalamic-pituitary axis; abrupt cessation may lead to fatigue, weight loss, and increased fracture risk.

Contraindications

Certain individuals should refrain from using testosterone and anabolic steroids as it may exacerbate existing medical conditions, including:

• Allergic responses to the drug
• Male breast cancer
• Prostate cancer in males
• Pregnancy or breastfeeding in females
• Individuals with liver, kidney, or heart diseases

Side Effects

The potential side effects of testosterone include:

• Nausea and vomiting
• Abdominal discomfort and diarrhea
• Swelling
• Altered libido
• Headaches
• Acne and oily skin
• Mood swings, such as anger, depression, and insomnia
• Increased perspiration
• Hair loss
• Gynecomastia

In women, testosterone can induce virilizing effects, including:

• Deepened voice
• Hoarseness
• Increased body hair
• Enlarged clitoris
• Irregular menstrual cycles

Long-term use can result in estrogen conversion, leading to breast enlargement and fluid retention, often reversing upon discontinuation.

Overdose

Overdosing on testosterone undecanoate is unusual. Even doses as high as 400-600 mg/day typically yield minimal acute effects, though symptoms may include diarrhea or abdominal cramps. Consultation with a healthcare provider is advisable for any significant concerns.

Dosage

In clinical settings, testosterone undecanoate is not standardly used. It is available as a 40 mg oral pill or a 250 mg/ml injectable solution, with injections administered into the muscle every 7-12 days. While some bodybuilders opt for more frequent injections, such practices increase the risk of infection or abscess formation. Injection sites should be rotated, and injections should not be given in the arms or abdomen. Bodybuilders commonly administer 200-400 mg/week, allowing for gradual systemic absorption.

Control

Testosterone undecanoate is a controlled substance, categorized under Class 3 of the Controlled Substance Act, and is illegal to possess, distribute, or sell in the USA.

Detection

This anabolic steroid and its metabolites remain detectable in urine for up to 2-3 weeks post-injection, influencing bodybuilders’ preferences for off-season usage.

Availability

Most bodybuilders acquire testosterone undecanoate through illegal markets. It may be sourced from Europe, Japan, Mexico, Spain, Brazil, and Thailand, though product quality remains highly variable. Prices typically range from $60-$100 for approximately 50 pills (40 mg each). Quality control is often lacking, with counterfeit products prevalent.

Final Word

Andriol is generally considered a last-resort option for bodybuilders due to its scarcity, high cost, and questionable efficacy, making it likely that users will encounter counterfeit versions.